|4-((6S,9S,9aS)-1-(苄基氨甲酰)-2,9-二甲基-4,7-二氧-8-(喹啉-8-基甲基)八氢-2H-吡嗪并[2,1-c][1,2,4]三嗪-6-基)甲基)苯基磷酸二氢单酯|CsnPharm

CAS No.: 1422253-38-0

4-(((6S,9S,9aS)-1-(Benzylcarbamoyl)-2,9-dimethyl-4,7-dioxo-8-(quinolin-8-ylmethyl)octahydro-2H-pyrazino[2,1-c][1,2,4]triazin-6-yl)methyl)phenyl dihydrogen phosphate Catalog No. CSN22491

Synonyms: C-82 prodrug;ICG-001 analog;foscenvivint

PRI-724 is a selective inhibitor of the CBP/β-catenin interaction.

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靶点选择性

生物活性

实验方案

技术信息

生物活性

描述PRI-724 is a selective inhibitor of the CBP/β-catenin interaction.
临床研究

NCT号	适应症或疾病	临床期	招募状态	预计完成时间	地点
NCT01606579	Acute Myeloid Leukemia ... more >> Chronic Myeloid Leukemia Collapse <<	Phase 1 Phase 2	Completed	-	United States, Georgia ... more >> Emory University / Winship Cancer Institute Atlanta, Georgia, United States, 30322 United States, Massachusetts University of Massachusetts Medical Center Worcester, Massachusetts, United States, 01655 United States, New Mexico New Mexico Cancer Care Alliance Albuquerque, New Mexico, United States, 87106 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27710 United States, Ohio Ohio State University Columbus, Ohio, United States, 43210-1267 United States, Texas University of Texas M.D. Anderson Cancer Center Houston, Texas, United States, 77030 Collapse <<
NCT02195440	Hepatitis C Virus-infected Cir... more >>rhosis Collapse <<	Phase 1	Completed	-	Japan ... more >> Tokyo metropolitan Komagome Hospital Tokyo, Japan Collapse <<
NCT02413853	Colorectal Adenocarcinoma ... more >> Stage IVA Colorectal Cancer Stage IVB Colorectal Cancer Collapse <<	Phase 2	Withdrawn(Study drug supply is... more >>sues) Collapse <<	November 2018	United States, California ... more >> USC Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 Collapse <<

实验方案

计算器摩尔计算器总药量计算器工作液计算器
储存液制备
- 1 mg
- 5 mg
- 10 mg
- 1 mM
- 1.5183 mL
- 7.5914 mL
- 15.1828 mL
- 5 mM
- 0.3037 mL
- 1.5183 mL
- 3.0366 mL
- 10 mM
- 0.1518 mL
- 0.7591 mL
- 1.5183 mL

技术信息

CAS号

1422253-38-0

储存条件

粉末: Sealed in dry,2-8°C

液体: -20°C:3-6 月 -80°C:12月

分子式

C33H35N6O7P

运输

蓝冰

分子量

658.64

别名

C-82 prodrug;ICG-001 analog;foscenvivint

溶解度

DMSO	100.0 mg/mL (151.8 mM)
Water	Insoluble
Ethanol	2.0 mg/mL (3.0 mM)

动物实验配方

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NCT号	适应症或疾病	临床期	招募状态	预计完成时间	地点

NCT01606579	Acute Myeloid Leukemia ... more >> Chronic Myeloid Leukemia Collapse <<	Phase 1 Phase 2	Completed	-	United States, Georgia ... more >> Emory University / Winship Cancer Institute Atlanta, Georgia, United States, 30322 United States, Massachusetts University of Massachusetts Medical Center Worcester, Massachusetts, United States, 01655 United States, New Mexico New Mexico Cancer Care Alliance Albuquerque, New Mexico, United States, 87106 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27710 United States, Ohio Ohio State University Columbus, Ohio, United States, 43210-1267 United States, Texas University of Texas M.D. Anderson Cancer Center Houston, Texas, United States, 77030 Collapse <<
NCT02195440	Hepatitis C Virus-infected Cir... more >>rhosis Collapse <<	Phase 1	Completed	-	Japan ... more >> Tokyo metropolitan Komagome Hospital Tokyo, Japan Collapse <<
NCT02413853	Colorectal Adenocarcinoma ... more >> Stage IVA Colorectal Cancer Stage IVB Colorectal Cancer Collapse <<	Phase 2	Withdrawn(Study drug supply is... more >>sues) Collapse <<	November 2018	United States, California ... more >> USC Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 Collapse <<
NCT02828254	-	-	Completed	-	Japan ... more >> Tokyo metropolitan Komagome Hospital Tokyo, Japan Collapse <<
NCT01764477	Advanced Pancreatic Cancer ... more >> Metastatic Pancreatic Cancer Pancreatic Adenocarcinoma Collapse <<	Phase 1	Completed	-	United States, California ... more >> USC Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 University of California, San Francisco San Francisco, California, United States, 94115 United States, Massachusetts Massachusetts General Hospital Cancer Center Boston, Massachusetts, United States, 02114 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, Washington University of Washington Seattle Cancer Care Alliance Seattle, Washington, United States, 98109 Collapse <<
NCT03620474	Hepatitis C H... more >>epatitis B Liver Cirrhoses Collapse <<	Phase 1 Phase 2	Recruiting	July 2020	Japan ... more >> Tokyo Metropolitan Komagome Hospital Recruiting Bunkyō-Ku, Tokyo, Japan, 113-8677 Contact: Kiminori Kimura +81-3-3823-2101 kkimura@cick.jp Contact: Akemi Ikoma +81-3-3823-2101 ikomaakm@cick.jp Collapse <<
NCT01302405	Advanced Solid Tumors	Phase 1	Terminated(closing due to low ... more >>enrollment, no safety issues) Collapse <<	-	United States, Arizona ... more >> Mayo Clinic Scottsdale, Arizona, United States, 85259-5499 United States, California University of Southern California, Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 United States, Minnesota Mayo Clinic, Department of Oncology Rochester, Minnesota, United States, 55901 Collapse <<

4-(((6S,9S,9aS)-1-(Benzylcarbamoyl)-2,9-dimethyl-4,7-dioxo-8-(quinolin-8-ylmethyl)octahydro-2H-pyrazino[2,1-c][1,2,4]triazin-6-yl)methyl)phenyl dihydrogen phosphate Catalog No. CSN22491

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